Apitolisib (Synonyms: GDC-0980; GNE 390; RG 7422)

CAS NO.:1032754-93-0

Molecular Formula:C₂₃H₃₀N₈O₃S

Molecular Weight:498.6011

Purity: > 98%

Solubility (R.T.: 25℃): DMSO

Stability: - 20℃ 2 years

Apitolisib (GDC-0980, RG7422) is a potent, class I PI3K inhibitor for PI3Kα/β/δ/γ with IC50 of 5 nM/27 nM/7 nM/14 nM in cell-free assays, respectively. Also a mTOR inhibitor with Ki of 17 nM in a cell-free assay, and highly selective versus other PIKK family kinases. Phase 2.

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