cis-Pralsetinib (cis-BLU-667)

CAS NO.:2097132-93-7

Molecular Formula:C₂₇H₃₂FN₉O₂

Molecular Weight:533.60

Purity: > 98%

Solubility (R.T.: 25℃): DMSO

Stability: - 20℃ 2 years

cis-Pralsetinib (cis-BLU-667) is a highly potent and selective inhibitor of rearranged during transfection (RET), with IC50s ranging from 0.3 to 0.4 nM for WT RET and four enzyme variants (V804L, V804M, M918T, CCDC6-RET), and with broad, robust and anti-tumor activity against multiple RET-driven solid tumor types.

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Quality Control by H-NMR,C-NMR,LC-MS,HPLC.

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