R10130 |
VX-680 (Tozasertib, MK-0457) |
VX-680 (Tozasertib, MK-0457) is a pan-Aurora inhibitor, mostly against Aurora A
|
R10131 |
Momelotinib (CYT387) |
Momelotinib (CYT387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 1
|
R10132 |
Canagliflozin |
Canagliflozin is a highly potent and selective SGLT2 inhibitor for hSGLT2 with I
|
R10136 |
Torkinib;PP242 |
Torkinib (PP242) is a selective mTOR inhibitor with IC50 of 8 nM in cell-free as
|
R10137 |
AP23464 |
CAS NO.:845895-51-4Product Name:AP-23464Synonyms:EINEC:Molecular Formula:C26H30N
|
R10138 |
Tivozanib;AV-951; KRN951 |
Tivozanib (AV-951) is a potent and selective VEGFR inhibitor for VEGFR1/2/3 with
|
R10139 |
Roscovitine; Seliciclib |
Roscovitine (Seliciclib, CYC202) is a potent and selective CDK inhibitor for Cdc
|
R10140 |
Daclatasvir dihydrochloride (BMS-790052 dihydrochloride) |
Daclatasvir (BMS-790052) is a highly selective inhibitor of HCV NS5A with EC50 o
|
R10141 |
SB705498 |
SB705498 is a TRPV1 antagonist for hTRPV1, antagonizes capsaicin, acid, and heat
|
R10143 |
Cabozantinib (XL184; BMS-907351) |
Cabozantinib (XL184, BMS-907351) is a potent VEGFR2 inhibitor with IC50 of 0.035
|
R10145 |
ABT102 |
CAS NO.:808756-71-0Product Name:ABT-102Synonyms:ABT-102;1-[(1R)-5-tert-butyl-2,3
|
R10146 |
XL765 |
Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ
|
R10147 |
LY335979 |
Zosuquidar (LY335979) is a potent modulator of P-glycoprotein-mediated multi-dru
|
R10149 |
Ticagrelor (AZD6140; AR-C 126532XX) |
Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist with K
|
R10150 |
Ceritinib; LKD378 |
Ceritinib (LDK378) is potent inhibitor against ALK with IC50 of 0.2 nM in cell-f
|
R10151 |
E7080; Lenvatinib |
Lenvatinib (E7080) is a multi-target inhibitor, mostly for VEGFR2(KDR)/VEGFR3(Fl
|
R10152 |
Neratinib; HKI272 |
Neratinib (HKI-272) is a highly selective HER2 and EGFR inhibitor with IC50 of 5
|
R10153 |
Roxadustat (FG-4592) |
Roxadustat (FG-4592) is an HIF α prolyl hydroxylase inhibitor in a cell-free ass
|
R10154 |
CTP518 |
|
R10155 |
Posaconazole; SCH56592; Noxafil |
Posaconazole is a sterol C14ɑ demethylase inhibitor with an IC50 of 0.25 nM.
|
R10156 |
Nintedanib; BIBF1120 |
Nintedanib (BIBF 1120) is a potent triple angiokinase inhibitor for VEGFR1/2/3,
|
R10157 |
AZD9291 Intermediate1 |
Osimertinib (AZD9291) is an oral, irreversible, and mutant-selective EGFR inhibi
|
R10158 |
AZD9291 Intermediate2 |
Osimertinib (AZD9291) is an oral, irreversible, and mutant-selective EGFR inhibi
|
R10159 |
Anacetrapib; MK0859 |
Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C
|
R10160 |
Omarigliptin; MK3102 |
Omarigliptin(MK-3102) is a potent, selective and long-acting DPP-4 inhibitor wit
|