R10009 |
AZD8055 |
AZD8055 is a novel ATP-competitive mTOR inhibitor with IC50 of 0.8 nM in MDA-MB-
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R10011 |
BIO-acetoxime; GSK3 Inhibitor IX |
BIO-acetoxime is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fol
|
R10013 |
PF 04691502 |
PF-04691502 is an ATP-competitive PI3K(α/β/δ/γ)/mTOR dual inhibitor with Ki of 1
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R10014 |
AKT inhibitor VIII (AKTI-1/2) |
CAS NO.:612847-09-3Product Name:1-(1-(4-(6-Phenyl-1H-imidazo[4,5-g]quinoxalin-7-
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R10027 |
KU-0063794 |
KU-0063794 is a potent and highly specific dual-mTOR inhibitor of mTORC1 and mTO
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R10040 |
IP-145; Duvelisib; INK1197 |
Duvelisib (IPI-145, INK1197) is a novel and selective PI3K δ/γ inhibitor with Ki
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R10044 |
WZ4003 |
WZ4003 is a highly specific NUAK kinase inhibitor with IC50 of 20 nM and 100 nM
|
R10072 |
GSK690693 |
GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM
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R10073 |
Apitolisib (Synonyms: GDC-0980; GNE 390; RG 7422) |
Apitolisib (GDC-0980, RG7422) is a potent, class I PI3K inhibitor for PI3Kα/β/δ/
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R10079 |
GSK2636771 |
GSK2636771 is a potent, orally bioavailable, PI3Kβ-selective inhibitor, sensitiv
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R10082 |
Palomid 529; P529 |
Palomid 529 (P529) inhibits both the mTORC1 and mTORC2 complexes, reduces phosph
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R10085 |
KU-55933 |
KU-55933 (ATM Kinase Inhibitor) is a potent and specific ATM inhibitor with IC50
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R10092 |
TWS11 |
TWS119 is a GSK-3β inhibitor with IC50 of 30 nM in a cell-free assay; capable of
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R10107 |
NVPBKM120 |
BKM120 (NVP-BKM120, Buparlisib) is a selective PI3K inhibitor of p110α/β/δ/γ wit
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R10136 |
Torkinib;PP242 |
Torkinib (PP242) is a selective mTOR inhibitor with IC50 of 8 nM in cell-free as
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R10146 |
XL765 |
Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ
|
R10167 |
PI103 Free base |
PI-103 is a multi-targeted PI3K inhibitor for p110α/β/δ/γ with IC50 of 2 nM/3 nM
|
R10168 |
YM201636 |
YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p11
|
R10180 |
Torin2 |
Torin 2 is a potent and selective mTOR inhibitor with IC50 of 0.25 nM in p53−/−
|
R10210 |
BYL719 |
Alpelisib (BYL719) is a potent and selective PI3Kα inhibitor with IC50 of 5 nM i
|
R10243 |
GDC0941; Pictilisib |
Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM in cell
|
R10343 |
Bikinin; Abrasin |
Bikinin is an ATP-competitive Arabidopsis GSK-3 inhibitor, and acts as a strong
|
R10373 |
GDC0941 |
Pictilisib (GDC-0941) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM in cell
|
R10486 |
TEPP46; ML265 |
TEPP-46 is a potent and selective activator of recombinant pyruvate kinase M2 (P
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R10493 |
AKT inhibitor IV |
|