R10332 |
Molibresib (Synonyms: GSK 525762A; I-BET 762) |
Molibresib (GSK 525762A; I-BET 762) is a BET bromodomain inhibitor with IC50 of
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R10349 |
AMI-1 |
AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor with IC
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R10369 |
GSK126 |
GSK126 is a potent, highly selective EZH2 methyltransferase inhibitor with IC50
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R10372 |
Baricitinib (INCB28050, LY3009104) |
Baricitinib (LY3009104, INCB028050) is a selective JAK1 and JAK2 inhibitor with
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R10374 |
Ruxolitinib phosphate;INCB018424 phosphate |
Ruxolitinib (INCB018424) is the first potent, selective, JAK1/2 inhibitor to ent
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R10409 |
(+)-JQ1 |
(+)-JQ1 is a BET bromodomain inhibitor, with IC50 of 77 nM/33 nM for BRD4(1/2) i
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R10422 |
BRD73954 |
BRD73954 is a potent and selective HDAC inhibitor with IC50 of 36 nM and 120 nM
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R10424 |
JNJ26481585; Quisinostat |
Quisinostat is an orally available, potent, hydroxamate, pan-HDACi with broad ac
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R10494 |
Tasocitinib; CP-690550 |
Tofacitinib (CP-690550,Tasocitinib) is a novel inhibitor of JAK3 with IC50 of 1
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R10516 |
Decitabine; NSC127716 |
Decitabine is a potent inhibitor of DNA methylation, used to treat myelodysplast
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R10536 |
Tofacitinib citrate (Tasocitinib citrate; CP-690550 citrate) |
Tofacitinib (CP-690550) Citrate is a novel inhibitor of JAK3 with IC50 of 1 nM i
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R10568 |
Fedratinib; TG101348 |
Fedratinib (SAR302503, TG101348) is a selective inhibitor of JAK2 with IC50 of 3
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R10572 |
Belinostat;PXD101 |
Belinostat (PXD101) is a novel HDAC inhibitor with IC50 of 27 nM in a cell-free
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R10617 |
Pracinostat (SB939) |
Pracinostat (SB939) is a potent pan-HDAC inhibitor with IC50 of 40-140 nM with e
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R10621 |
JW55 |
JW 55 is an inhibitor of the PARP domain of tankyrase 1 and 2 (TNKS1/2).
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R10669 |
TMP269 |
TMP269 is a potent, selective class IIa HDAC inhibitor with IC50 of 157 nM, 97 n
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R10671 |
NexturastatA |
Nexturastat A is a potent and selective HDAC6 inhibitor with IC50 of 5 nM, >1
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R10673 |
NSC 42834;JAK2 Inhibitor V; Z3 |
Z3 is a novel specific inhibitor of Jak2 tyrosine kinase.
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R10681 |
NSC693627; AC1O75RE; JIB04; FD5031; NSC-693627 |
JIB-04 is a pan-selective Jumonji histone demethylase inhibitor with IC50 of 230
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R10697 |
HDAC-IN-7 (Chidamide impurity) |
Chidamide(CS055; HBI-8000) is a class I HDAC inhibitor with IC50s of 95/160/67/7
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R10702 |
RG108;N-Phthalyl-L-tryptophan |
RG108 is an inhibitor of DNA methyltransferase with IC50 of 115 nM in a cell-fre
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R10709 |
JANEX-1 (Synonyms: WHI-P131; Jak3 inhibitor I) |
Janex-1 is a cell-permeable, reversible, potent, ATP-competitive, and specific i
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R10710 |
WHI-P180 |
WHI-P180 (Janex 3) is a multi-kinase inhibitor; inhibits RET, KDR and EGFR with
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R10732 |
MC1568 |
MC1568 is a selective HDAC inhibitor for maize HD1-A with IC50 of 100 nM in a ce
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R10759 |
CAY10683;Santacruzamate A |
Santacruzamate A (CAY10683) is a potent and selective HDAC inhibitor with IC50 o
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