R10202 |
AZD4547 |
AZD4547 is a novel selective FGFR inhibitor targeting FGFR1/2/3 with IC50 of 0.2
|
R10233 |
Tyrphostin A9;Tyrphostin 9; Malonoben |
Tyrphostin 9 is firstly designed as an EGFR inhibitor with IC50 of 460 μM, but i
|
R10235 |
GSK1838705A |
GSK1838705A is a potent and reversible IGF-IR and the insulin rec
|
R10253 |
Dacomitinib,PF299804 |
Dacomitinib (PF299804, PF299) is a potent, irreversible pan-ErbB inhibitor, most
|
R10254 |
AZD9291 Mesylate |
AZD-9291 is a potent and selective mutated forms EGFR inhibitor(Exon 19 deletion
|
R10255 |
LY2874455; dovitinib |
LY2874455 is a pan-FGFR inhibitor with IC50 of 2.8 nM, 2.6 nM, 6.4 nM, and 6 nM
|
R10256 |
Blu9931 |
BLU9931 is a potent, highly selective, and irreversible fibroblast growth factor
|
R10259 |
AG490 |
AG-490 (Tyrphostin B42) is an inhibitor of EGFR with IC50 of 0.1 μM in cell-free
|
R10283 |
Nintedanib esylate; BIBF1120 esylate |
Nintedanib (BIBF 1120) is a potent triple angiokinase inhibitor for VEGFR1/2/3,
|
R10296 |
Afatinib; BIBW2992 |
Afatinib (BIBW2992) irreversibly inhibits EGFR/HER2 including EGFR(wt), EGFR(L85
|
R10331 |
Cabozantinib S-malate (XL184 S-malate; BMS-907351 S-malate) |
abozantinib malate (XL184) is the malate of Cabozantinib, a potent VEGFR2 inhibi
|
R10339 |
PLX-3397; Pexidartinib |
Pexidartinib (PLX3397) is an oral, potent mutil-targeted receptor tyrosine kinas
|
R10358 |
Nintedanib; BIBF1120; Vargatef |
Nintedanib (BIBF 1120) is a potent triple angiokinase inhibitor for VEGFR1/2/3,
|
R10448 |
Imatinib; STI571 |
Imatinib (STI571) is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC5
|
R10449 |
Gefitinib; ZD1839 |
Gefitinib (ZD-1839) is an EGFR inhibitor for Tyr1173, Tyr992, Tyr1173 and Tyr992
|
R10514 |
Axitinib; AG013736 |
Axitinib is a multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFRβ and c-Kit
|
R10535 |
Afatinib dimaleate; BIBW2992 dimaleate |
Afatinib (BIBW2992) Dimaleate irreversibly inhibits EGFR/HER2 including EGFR(wt)
|
R10540 |
Regorafenib monohydrate |
Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFR??, Kit
|
R10545 |
CANGRELOR |
Regorafenib is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFR, Kit,
|
R10569 |
Pelitinib |
Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM
|
R10585 |
AZD3759 |
AZD3759 is a potent, oral active, central nervous system-penetrant, EGFR inhibit
|
R10699 |
AG18 |
AG-18 inhibits EGFR with IC50 of 35 μM.
|
R10711 |
AG-1517 |
PD153035 HCl is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2
|
R10727 |
Quizartinib;AC-220 |
Quizartinib (AC220) is a second-generation FLT3 inhibitor for Flt3(ITD/WT) with
|
R10733 |
Semaxinib;SU5416 |
Semaxanib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor with IC5
|