R10785 |
Savolitinib (Volitinib; HMPL-504; AZD-6094) |
Savolitinib(Volitinib; AZD-6094; Volitinib) is an orally bioavailable inhibitor
|
R10818 |
Varlitinib; ARRY 543 |
Varlitinib is a selective and potent ErbB1(EGFR) and ErbB2(HER2) inhibitor with
|
R10837 |
INCB28060 |
Capmatinib (INCB28060) is a novel, ATP-competitive inhibitor of c-MET with IC50
|
R10880 |
Lapatinib (GW572016; GW2016) |
Lapatinib, used in the form of Lapatinib Ditosylate, is a potent EGFR and ErbB2
|
R10867 |
LDC1267 |
LDC1267 is a highly selective TAM kinase inhibitor with IC50 of <5 nM, 8 nM,
|
R10881 |
Sorafenib (Synonyms: Bay 43-9006) |
Sorafenib (Bay 43-9006) is a potent, orally active multikinase inhibitor with IC
|
R10882 |
Sunitinib (Synonyms: SU 11248) |
Sunitinib Malate is a multi-targeted RTK inhibitor targeting VEGFR2 (Flk-1) and
|
R10891 |
Vatalanib |
Vatalanib (PTK787) 2HCl is an inhibitor of VEGFR2/KDR with IC50 of 37 nM in a ce
|
R10898 |
Lorlatinib (Synonyms: PF-06463922) |
PF-06463922 is a potent, dual ALK/ROS1 inhibitor with Ki of <0.02 nM, <0.0
|
R10900 |
CL-387785 ; EKI-785 |
CL-387785(EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFR with IC50 of
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R10904 |
Irbinitinib; ARRY-380; ONT-380 |
Irbinitinib(ARRY-380; ONT-380) is a potent and selective HER2 inhibitor with IC5
|
R10930 |
Icotinib |
Icotinib is a potent and specific EGFR inhibitor with IC50 of 5 nM, including th
|
R10941 |
Alectinib(CH5424802; RO5424802; AF802) |
Alectinib (CH5424802) is a potent ALK inhibitor with IC50 of 1.9 nM in cell-free
|
R11470 |
Apatinib methanesulfonate |
Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM
|
R11479 |
Lapatinib ditosylate;GW572016 ditosylate; GW2016 ditosylate |
Lapatinib, used in the form of Lapatinib Ditosylate, is a potent EGFR and ErbB2
|
R11514 |
Pazopanib (Synonyms: GW786034) |
Pazopanib is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FG
|
R11523 |
BMS-794833 |
BMS-794833 is a potent ATP competitive inhibitor of Met/VEGFR2 with IC50 of 1.7
|
R11536 |
PD168393 |
PD168393 is an irreversible EGFR inhibitor with IC50 of 0.70 nM, irreversibly al
|
R11550 |
Dovitinib |
Dovitinib (TKI258) Lactate is the Lactate of Dovitinib, which is a multitargeted
|
R11552 |
BFH-772 |
BFH772 is a novel potent oral VEGFR2 inhibitor, targeting VEGFR2 kinase with IC5
|
R11557 |
CH5183284; Debio 1347 |
CH5183284 is a selective and orally available FGFR inhibitor with IC50 of 9.3 nM
|
R11600 |
Bemcentinib (Synonyms: R428; BGB324) |
R428 (BGB324) is an inhibitor of Axl with IC50 of 14 nM, >100-fold selective
|
R11603 |
WZ3146 |
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and
|
R190306 |
AST2818 mesylate |
AST2818 mesylate is an EGFR inhibitor.
|
R2032681 |
BMS599626 |
BMS-599626 (AC480) is a selective and orally bioavailable HER1 and HER2 inhibito
|