R10006 |
Allitinib tosylate (Synonyms: AST-1306 (TsOH))/897383-62-9 Free base |
AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM
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R10042 |
CO1686; Rociletinib |
Rociletinib (CO-1686, AVL-301) is an irreversible, mutant-selective EGFR inhibit
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R10087 |
AZD9291 |
Osimertinib (AZD9291) is an oral, irreversible, and mutant-selective EGFR inhibi
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R10126 |
WZ4002 |
WZ4002 is a novel, mutant-selective EGFR inhibitor for EGFR(L858R)/(T790M) with
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R10152 |
Neratinib; HKI272 |
Neratinib (HKI-272) is a highly selective HER2 and EGFR inhibitor with IC50 of 5
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R10233 |
Tyrphostin A9;Tyrphostin 9; Malonoben |
Tyrphostin 9 is firstly designed as an EGFR inhibitor with IC50 of 460 μM, but i
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R10253 |
Dacomitinib,PF299804 |
Dacomitinib (PF299804, PF299) is a potent, irreversible pan-ErbB inhibitor, most
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R10254 |
AZD9291 Mesylate |
AZD-9291 is a potent and selective mutated forms EGFR inhibitor(Exon 19 deletion
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R10259 |
AG490 |
AG-490 (Tyrphostin B42) is an inhibitor of EGFR with IC50 of 0.1 μM in cell-free
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R10449 |
Gefitinib; ZD1839 |
Gefitinib (ZD-1839) is an EGFR inhibitor for Tyr1173, Tyr992, Tyr1173 and Tyr992
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R10569 |
Pelitinib |
Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM
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R10585 |
AZD3759 |
AZD3759 is a potent, oral active, central nervous system-penetrant, EGFR inhibit
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R10699 |
AG18 |
AG-18 inhibits EGFR with IC50 of 35 μM.
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R10711 |
AG-1517 |
PD153035 HCl is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2
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R10818 |
Varlitinib; ARRY 543 |
Varlitinib is a selective and potent ErbB1(EGFR) and ErbB2(HER2) inhibitor with
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R10880 |
Lapatinib (GW572016; GW2016) |
Lapatinib, used in the form of Lapatinib Ditosylate, is a potent EGFR and ErbB2
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R10900 |
CL-387785 ; EKI-785 |
CL-387785(EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFR with IC50 of
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R10904 |
Irbinitinib; ARRY-380; ONT-380 |
Irbinitinib(ARRY-380; ONT-380) is a potent and selective HER2 inhibitor with IC5
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R10930 |
Icotinib |
Icotinib is a potent and specific EGFR inhibitor with IC50 of 5 nM, including th
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R11536 |
PD168393 |
PD168393 is an irreversible EGFR inhibitor with IC50 of 0.70 nM, irreversibly al
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R11603 |
WZ3146 |
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and
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R190306 |
AST2818 mesylate |
AST2818 mesylate is an EGFR inhibitor.
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R2032681 |
BMS599626 |
BMS-599626 (AC480) is a selective and orally bioavailable HER1 and HER2 inhibito
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R2032738 |
AV412 |
AV-412 free base (MP-412 free base) is an EGFR inhibitor with IC50s of 0.75, 0.5
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