R10091 |
LCZ696;Sacubitril;Valsartan |
Varespladib (LY315920) is a potent and selective human non-pancreatic secretory
|
R10112 |
Abiraterone Acetate; CB7630 |
Abiraterone Acetate is an acetate salt form of Abiraterone which is a steroidal
|
R10113 |
Abiraterone; CB7598 |
Abiraterone is a potent CYP17 inhibitor with IC50 of 2 nM in a cell-free assay.
|
R10125 |
TOK001; VN1241 |
Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist
|
R10159 |
Anacetrapib; MK0859 |
Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C
|
R10162 |
Apremilast; CC10004 |
Apremilast (CC-10004) is a potent and orally active PDE4 and TNF-α inhibitor wit
|
R10209 |
indisulam; E7070 |
Indisulam (E7070) is a carbonic anhydrase inhbitor, is also a novel synthetic su
|
R10344 |
GW9662 |
GW9662 is a selective PPAR antagonist for PPARγ with IC50 of 3.3 nM in a cell-fr
|
R10432 |
Rivaroxaban; Xarelto; BAY 59-7939 |
Rivaroxaban is a direct inhibitor of Factor Xa with Ki and IC50 of 0.4 nM and 0.
|
R10444 |
Olprinone |
Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.
|
R10456 |
Gimeracil |
Gimeracil is an inhibitor of dihydropyrimidine dehydrogenase, which inhibits the
|
R10482 |
Tadalafil |
Tadalafil is a PDE-5 inhibitor with IC50 of 1.8 nM in a cell-free assay.
|
R10485 |
Epacadostat (Synonyms: INCB 024360) |
Epacadostat (INCB024360) is a potent and selective indoleamine 2,3-dioxygenase (
|
R10526 |
Anagrelide hydrochloride; BL4162A |
Anagrelide is a drug used for the treatment of essential thrombocytosis.
|
R10570 |
Safinamide mesylate |
Safinamide Mesylate is mesylate salt of Safinamide, selectively and reversibly i
|
R10591 |
NSC14613; PluriSln1 |
PluriSIn1 is an inhibitor of the stearoyl-coA desaturase 1 (SCD1), which is able
|
R10632 |
AGI-6780 |
AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 2
|
R10648 |
Dimethyloxaloylglycine;DMOG |
DMOG is an antagonist of α-ketoglutarate cofactor and inhibitor for HIF prolyl h
|
R10659 |
Fenretinide; 4-HPR |
Fenretinide is a synthetic retinoid agonist. It is an antiproliferative, antioxi
|
R10724 |
Moclobemide |
Moclobemide is a MAO-A (5-HT) inhibitor with IC50 of 6.1 μM.
|
R10735 |
U-104 |
U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with Ki
|
R10801 |
Deltarasin |
Deltarasin is a small molecular inhibitor of KRAS-PDEδ interaction with Kd of 38
|
R10665 |
IDO-IN-7;NLG-919 analogue; GDC-0919 analogue |
NLG919 is a potent IDO (indoleamine-(2,3)-dioxygenase) pathway inhibitor with Ki
|
R10842 |
Mycophenolate mofetil; Linfonex |
Mycophenolate Mofetil is a non-competitive, selective and reversible inhibitor o
|
R10841 |
Mycophenolic acid |
Mycophenolic acid is a potent IMPDH inhibitor and the active metabolite of an im
|